Talazoparib

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Molecule Structure

Scientific Name

Talazoparib

Description of the Drug

Talazoparib is a poly-ADP ribose polymerase inhibitor used to treat HER2-, BRCA mutated locally advanced or metastatic breast cancer.

Source: DrugBank Online – DrugBank.com. Retrieved 2023-03-10 from
http://www.drugbank.ca/drugs/DB11760

Brand Name(s)

Not Available

Company Owner(s)

Pfizer Inc

Mechanism(s) Of Action

Target Name Target Type Action Type Target ChEMBL ID
Poly [ADP-ribose] polymerase-1 SINGLE PROTEIN INHIBITOR CHEMBL3105
Poly [ADP-ribose] polymerase 2 SINGLE PROTEIN INHIBITOR CHEMBL5366

Unichem Links

SureChEMBL SCHEMBL2299348
DrugBank DB11760
PubChem: Thomson Pharma 89447774
PubChem 135565082
Nikkaji J3.353.317I
PDBe 2YQ
BindingDB 50084621
DrugCentral 5300
ChemicalBook CB22615112
rxnorm TALZENNA TALAZOPARIB TALAZOPARIB TOSYLATE
ZINC ZINC000072318110