Lorlatinib
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Scientific Name
Lorlatinib
Description of the Drug
Lorlatinib is an anaplastic lymphoma kinase inhibitor used to treat anaplastic lymphoma kinase positive metastatic non small cell lung cancer.
Source: DrugBank Online – DrugBank.com. Retrieved 2023-03-10 from
http://www.drugbank.ca/drugs/DB12130
http://www.drugbank.ca/drugs/DB12130
Brand Name(s)
Lorbrena
Company Owner(s)
Pfizer Inc
Mechanism(s) Of Action
Target Name | Target Type | Action Type | Target ChEMBL ID |
---|---|---|---|
ALK tyrosine kinase receptor | SINGLE PROTEIN | INHIBITOR | CHEMBL4247 |
EML4-ALK | CHIMERIC PROTEIN | INHIBITOR | CHEMBL3883330 |
Clinical Trial(s)
Unichem Links
SureChEMBL | SCHEMBL15261807 | |
DrugBank | DB12130 | |
PubChem | 71731823 | |
Nikkaji | J3.339.850F | |
PDBe | 5P8 | |
BindingDB | 50018830 | |
DrugCentral | 5302 | |
ChemicalBook | CB02716543 | |
Guide to Pharmacology | 7476 | |
rxnorm | LORBRENA | LORLATINIB |
ChEBI | 143117 | |
ZINC | ZINC000098208524 |