Gilteritinib

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Molecule Structure

Scientific Name

Gilteritinib

Description of the Drug

Gilteritinib is an AXL receptor tyrosine kinase inhibitor used to treat relapsed or refractory acute myeloid leukemia.

Source: DrugBank Online – DrugBank.com. Retrieved 2023-03-10 from
http://www.drugbank.ca/drugs/DB12141

Brand Name(s)

Not Available

Company Owner(s)

Astellas Pharma Us Inc

Mechanism(s) Of Action

Target Name Target Type Action Type Target ChEMBL ID
Tyrosine-protein kinase receptor UFO SINGLE PROTEIN INHIBITOR CHEMBL4895
Tyrosine-protein kinase receptor FLT3 SINGLE PROTEIN INHIBITOR CHEMBL1974

Unichem Links

SureChEMBL SCHEMBL282229
Human Metabolome Database HMDB0252717
DrugBank DB12141
PubChem: Thomson Pharma 103775109
PubChem 49803313
Nikkaji J3.425.284J
PDBe C6F
BindingDB 144315
DrugCentral 5306
ChemicalBook CB82725626
Guide to Pharmacology 8708
rxnorm XOSPATA GILTERITINIB FUMARATE GILTERITINIB
ChEBI 145372
ZINC ZINC000113476229